1. 2019
  2. Neurotensin Analogues Containing Cyclic Surrogates of Tyrosine at Position 11 Improve NTS2 Selectivity Leading to Analgesia without Hypotension and Hypothermia

    Eiselt, E., Gonzalez, S., Martin, C., Chartier, M., Betti, C., Longpre, J-M., Cavelier, F., Tourwe, D., Gendron, L., Ballet, S. & Sarret, P., Nov 2019, In : ACS Chemical Neuroscience. 10, 11, p. 4535-4544

    Research output: Contribution to journalArticleResearchpeer-review

  3. Trifluoromethylated Proline Surrogates as Part of "Pro-Pro" Turn-Inducing Templates

    Gadais, C., Van holsbeeck, K., Moors, S. L. C., Buyst, D., Feher, K., Van Hecke, K., Tourwe, D., Brigaud, T., Martin, C., De Proft, F., Pytkowicz, J., Martins, J. C., Chaume, G. & Ballet, S., 15 Jul 2019, In : ChemBioChem. 20, 19, p. 2513-2518

    Research output: Contribution to journalArticleResearchpeer-review

  4. 2018
  5. Synthesis of novel arylazepinone dipeptide mimetics and 1,5-benzothiazepinones as local constraints in peptidomimetic design

    Van den Hauwe, R., Van der Poorten, O., Ballet, S., Eiselt, E., Sarret, P., Gendron, L. & Tourwe, D., Sep 2018, In : Journal of Peptide Science. 24, p. S120-S120

    Research output: Contribution to journalMeeting abstract (Journal)Research

  6. Trifluoromethylated proline surrogates as part of 'Pro-Pro' turn-inducing templates for the design of beta-hairpin mimetics.

    Gadais, C., Van Holsbeeck, K., Moors, S., Feher, K., Pytkowicz, J., Martins, J., De Proft, F., Tourwe, D., Brigaud, T., Martin, C., Chaume, G. & Ballet, S., Sep 2018, In : Journal of Peptide Science. 24, p. S117-S117

    Research output: Contribution to journalMeeting abstract (Journal)Research

  7. Synthesis and in Vitro Evaluation of Stabilized and Selective Neuromedin U-1 Receptor Agonists

    De Prins, A., Martin, C., Van Wanseele, Y., Tömböly, C., Tourwé, D., Caveliers, V., Holst, B., Van Eeckhaut, A., Rosenkilde, M. M., Smolders, I. & Ballet, S., 10 May 2018, In : ACS Medicinal Chemistry Letters. 9, 5, p. 496–501 6 p.

    Research output: Contribution to journalArticleResearchpeer-review

  8. Indoloazepinone-Constrained Oligomers as Cell-Penetrating and Blood-Brain-Barrier-Permeating Compounds

    Van der Poorten, O., Legrand, B., Vezenkov, L. L., Garcia-Pindado, J., Bettache, N., Knuhtsen, A., Pedersen, D. S., Sanchez-Navarro, M., Martinez, J., Teixido, M., Garcia, M., Tourwe, D., Amblard, M. & Ballet, S., 4 Apr 2018, In : ChemBioChem. 19, 7, p. 696-705 10 p.

    Research output: Contribution to journalArticleResearchpeer-review

  9. Discovery of potent NMUR1 selective Neuromedin U analogs with increased resistance against biodegradation

    De Prins, A., Martin, C., Van Wanseele, Y., Tömböly, C., Tourwe, D., Caveliers, V., Van Eeckhaut, A., Holst, B., Rosenkilde, M. M., Smolders, I. & Ballet, S., 28 Feb 2018, (Unpublished).

    Research output: Unpublished contribution to conferencePosterResearch

  10. Development of potent and proteolytically stable human neuromedin U receptor agonists

    De Prins, A., Martin, C., Van Wanseele, Y., Skov, L. J., Tömböly, C., Tourwe, D., Caveliers, V., Van Eeckhaut, A., Holst, B., Rosenkilde, M. M., Smolders, I. & Ballet, S., 20 Jan 2018, In : European Journal of Medicinal Chemistry. 144, p. 887-897 11 p.

    Research output: Contribution to journalArticleResearchpeer-review

  11. Rapid construction of substituted 3-amino-1,5-benzothiazepin-4(5H)-one dipeptide scaffolds through an Ugi-4CR - Ullmann cross-coupling sequence

    Van der Poorten, O., Van Den Hauwe, R., Hollanders, K., Tourwé, D., Jida, M. & Ballet, S., 1 Jan 2018, In : Organic & Biomolecular Chemistry. 16, 8, p. 1242-1246 5 p.

    Research output: Contribution to journalArticleResearchpeer-review

  12. Efficient One-Pot Access to Trisubstituted 2-Benzazepin-3-ones as Constrained Pseudopeptide Analogues and Privileged Scaffolds

    Van der Poorten, O., Jida, M., Tourwe, D. & Ballet, S., 2018, In : Current Medicinal Chemistry. 14, 4, p. 400-408 9 p.

    Research output: Contribution to journalArticleResearchpeer-review

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